Last Update: Sep 19, 2024
A Phase I, Open-label, Multi-center Study to Evaluate the Safety, Tolerability, Dosimetry, and Preliminary Activity of [177Lu]Lu-EVS459 in Patients With Ovarian and Lung Cancers
ClinicalTrials.gov Identifier:
Novartis Reference Number:CGIZ943A12101
All compounds are either investigational or being studied for (a) new use(s). Efficacy and safety have not been established. There is no guarantee that they will become commercially available for the use(s) under investigation.

Study Description

The purpose of this study is to evaluate the safety, tolerability, dosimetry and
preliminary efficacy of [177Lu]Lu-EVS459 and the safety and imaging properties of
[68Ga]Ga-EVS459 in patients aged ≥ 18 years with advanced high-grade serous ovarian
cancer (OC) or locally advanced unresectable or metastatic non-squamous non-small cell
lung carcinoma (non-sq. NSCLC). The study will be done in two parts. The first part is called "escalation" and the second
part is called "expansion". In both parts of the study, patients will initially be imaged
with a [68Ga]Ga EVS459 positron emission tomography (PET)/computed tomography (CT) or
PET/magnetic resonance imaging (MRI) scan. In the escalation part, different doses of
[177Lu]Lu-EVS459 will then be tested to identify recommended dose(s) (RD(s)) for further
evaluation. The expansion part of the study will examine the safety and preliminary
efficacy of [177Lu]Lu-EVS459 at the RD(s) determined during the escalation part. The end
of study will occur when at least 80% of the patients in the expansion part have
completed the follow-up for disease progression or discontinued from the study for any
reason, and all patients have completed treatment and the 36-month long-term follow-up
period.

Ovarian Cancer, Lung Cancer
Phase1
Recruiting
96
Sep 08, 2024
Aug 30, 2030
All
18 Years - 100 Years (Adult, Older Adult)

Interventions

Drug

[177Lu]Lu-EVS459

Radioligand therapy
Drug

[68Ga]Ga-EVS459

Radioligand imaging agent

Eligibility Criteria

Key Inclusion Criteria:

- Age >= 18 years old

- Patients with advanced high-grade serous ovarian cancer (OC) or locally advanced
unresectable or metastatic non-squamous non-small cell lung cancer (non sq. NSCLC)
with disease progression following, or intolerance to, at least 1 line of therapy

Key Exclusion Criteria:

- Absolute neutrophil count (ANC) < 1.5 x 10^9/L, hemoglobin < 10 g/dL, or platelet
count < 100 x 10^9/L

- QT interval corrected by Fridericia's formula (QTcF) ≥ 470 msec

- Creatinine clearance < 60 mL/min

- Unmanageable urinary tract obstruction or urinary incontinence

- Radiation therapy within 4 weeks prior to the first dose of [177Lu]Lu-EVS459

Other protocol-defined inclusion/exclusion criteria may apply.

Novartis Investigative Site

Recruiting

Tel Aviv,6423906,Israel

Worldwide Contacts

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Novartis Pharmaceuticals

Novartis Pharmaceuticals